Artigo Revisado por pares

Genetic Variants in Arachidonic Acid Pathway Genes Associated with NSAID-Exacerbated Respiratory Disease

2015; Future Medicine; Volume: 16; Issue: 8 Linguagem: Inglês

10.2217/pgs.15.43

ISSN

1744-8042

Autores

Pedro Ayuso, María del Carmen Plaza‐Seron, Natalia Blanca‐López, Inmaculada Doña, Paloma Campo, Gabriela Cantó, José Julio Laguna, Joan Bartra, Víctor Soriano, Miguel Blanca, J.A. Cornejo‐García, James R. Perkins,

Tópico(s)

Drug-Induced Adverse Reactions

Resumo

Aim: NSAIDs are the most frequent cause of hypersensitivity drug reactions. We have examined the association between NSAID-exacerbated respiratory disease (NERD) and genetic variants in arachidonic acid metabolism genes. Patients & methods: We included 250 NERD patients, 260 NSAID-tolerant asthmatic (NTA) subjects and 315 healthy controls. Results: Significant associations with NERD were identified for: ALOX15 rs3892408 C/C homozygous genotype (NERD vs NTA; p = 0.0001, pc = 0.0011; NERD vs controls; p = 0.0001, pc = 0.0011), PTGS-1 rs5789 A/A homozygous genotype (NERD vs NTA; p = 0.0001, pc = 0.0011; NERD vs controls; p = 0.0001, pc = 0.0011), PTGS-1 rs10306135 A/A homozygous genotype (NERD vs NTA; p = 0.0009, pc = 0.0091; NERD vs controls; p = 0.0064, pc = 0.045). Differences in ALOX5 copy number variations were also found (NERD vs NTA; p = 0.010; NERD vs controls; p = 0.0001). Conclusion: These results improve our understanding of the underlying mechanisms of NERD and may help develop a predictive test for this pathology. Original submitted 3 November 2014; Revision submitted 2 April 2015

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