Efficient Synthesis of 1-Sulfonyl-1,2,3-triazoles
2010; American Chemical Society; Volume: 12; Issue: 21 Linguagem: Inglês
10.1021/ol102087r
ISSN1523-7060
AutoresJessica Raushel, Valery V. Fokin,
Tópico(s)Sulfur-Based Synthesis Techniques
ResumoAn efficient room-temperature method for the synthesis of 1-sulfonyl-1,2,3-triazoles from in situ generated copper(I) acetylides and sulfonyl azides is described. The copper(I) thiophene-2-carboxylate (CuTC) catalyst produces the title compounds under both nonbasic anhydrous and aqueous conditions in good yields.
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