A convenient synthesis of L ‐1‐methylhistidine and L ‐1‐ethylhistidine

1972; Royal Netherlands Chemical Society; Volume: 91; Issue: 3 Linguagem: Inglês

10.1002/recl.19720910302

ISSN

1878-7096

Autores

H. C. Beyerman, L. Maat, A. van Zon,

Tópico(s)

Carbohydrate Chemistry and Synthesis

Resumo

Abstract Alkylation of the easily accessible methyl ester of L ‐ N a ,3‐dibenzoylhistidine with the aid of trimethyl‐ and triethyloxonium fluoroborate followed by decomposition with water and acid hydrolysis yielded L ‐1 ‐methyl‐ and L ‐1‐ethylhistidine respectively. Comparison with natural L ‐1‐methylhistidine confirmed the structure and optical purity.

Referência(s)