Discovery of potent, soluble and orally active TRPV1 antagonists. Structure–activity relationships of a series of isoxazoles
2011; Elsevier BV; Volume: 21; Issue: 15 Linguagem: Inglês
10.1016/j.bmcl.2011.01.051
ISSN1464-3405
AutoresPaul Ratcliffe, Lynn Abernethy, Nasrin Ansari, Ken Cameron, Tom Clarkson, Maureen Dempster, David A. Dunn, Anna-Marie Easson, Darren Edwards, Katy L. Everett, Helen Feilden, Koc-Kan Ho, Steve Kultgen, Peter Littlewood, John Maclean, Duncan McArthur, Deborah McGregor, Hazel McLuskey, Irina Neagu, Olaf Nimz, Lesley-Anne Nisbet, Michael Ohlmeyer, Ronnie Palin, Quynhchi Pham, Yajing Rong, Andrew L. Roughton, Melanie Sammons, R. N. Swanson, Heather Tracey, Glenn Walker,
Tópico(s)Bioactive Compounds and Antitumor Agents
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