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The influence of selective thromboxane synthetase inhibition with a novel imidazole derivative, UK-38,485, on prostanoid formation in man.

1983; Lippincott Williams & Wilkins; Volume: 68; Issue: 4 Linguagem: Inglês

10.1161/01.cir.68.4.821

1524-4539

Susan M. Fischer, Michael Struppler, B. Böhlig, C. Bernutz, W. Wober, Christian Weber,

Synthesis of β-Lactam Compounds

HomeCirculationVol. 68, No. 4The influence of selective thromboxane synthetase inhibition with a novel imidazole derivative, UK-38,485, on prostanoid formation in man. Free AccessAbstractPDF/EPUBAboutView PDFSections ToolsAdd to favoritesDownload citationsTrack citationsPermissions ShareShare onFacebookTwitterLinked InMendeleyReddit Jump toFree AccessAbstractPDF/EPUBThe influence of selective thromboxane synthetase inhibition with a novel imidazole derivative, UK-38,485, on prostanoid formation in man. S Fischer, M Struppler, B Böhlig, C Bernutz, W Wober and P C Weber S FischerS Fischer , M StrupplerM Struppler , B BöhligB Böhlig , C BernutzC Bernutz , W WoberW Wober and P C WeberP C Weber Originally published1 Oct 1983https://doi.org/10.1161/01.CIR.68.4.821Circulation. 1983;68:821–826 Previous Back to top Next FiguresReferencesRelatedDetailsCited By Sathler P, Santana M, Lourenço A, Rodrigues C, Abreu P, Cabral L and Castro H (2013) Human thromboxane synthase: comparative modeling and docking evaluation with the competitive inhibitors Dazoxiben and Ozagrel, Journal of Enzyme Inhibition and Medicinal Chemistry, 10.3109/14756366.2013.817403, 29:4, (527-531), Online publication date: 1-Aug-2014. Tanaka M, Ono K, Takegoshi T, Shiozawa T, Suzuki T, Nii S and Shibata H (2011) The Pharmacokinetics and Pharmacodynamics of a New Thromboxane Synthetase Inhibitor, 6-(1-Imidazolylmethyl)-5,6,7,8-tetrahydronaphthalene-2-carboxylic acid (DP-1904), in Man after Single Oral Administration, Journal of Pharmacy and Pharmacology, 10.1111/j.2042-7158.1989.tb06340.x, 41:10, (680-684), Online publication date: 12-Apr-2011. Carvalho M, Fortes Z, Nigro D, Oliveira M and Scivoletto R (2009) The Role of Thromboxane A 2 in the Altered Microvascular Reactivity in Two-Kidney, One-Clip Hypertension , Endothelium, 10.3109/10623329709053396, 5:3, (167-178), Online publication date: 1-Jan-1997. Dickinson R, Dack K, Steele J and Tute M (1996) Thromboxane modulating agents. 2. Thromboxane receptor antagonists derived from the thromboxane synthase inhibitor dazmegrel., Bioorganic & Medicinal Chemistry Letters, 10.1016/0960-894X(96)00299-5, 6:14, (1691-1696), Online publication date: 1-Jul-1996. 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October 1, 1983Vol 68, Issue 4 Advertisement Article InformationMetrics Copyright © 1983 by American Heart Associationhttps://doi.org/10.1161/01.CIR.68.4.821 Originally publishedOctober 1, 1983 PDF download Advertisement