Artigo Revisado por pares

Photochemical activation of trimethylsilylmethyl allylic sulfones for intramolecular 4+3 cycloaddition

1993; Elsevier BV; Volume: 34; Issue: 34 Linguagem: Inglês

10.1016/s0040-4039(00)73914-1

ISSN

1873-3581

Autores

Michael Harmata, Barry F. Herron,

Tópico(s)

Organic Chemistry Cycloaddition Reactions

Resumo

Irradiation of allylic sulfones 4–7 results in the formation of 4+3 cycloadducts 8–11. Although the yields are poor, this represents the first apparent photochemical generation of acyclic allylic cations for 4+3 cycloadditions. Mechanistically, this process is interpreted as an electron transfer process to form an internal radical cation/radical anion reactive intermediate. This eliminates p-tolylsulfinate anion to form an allylic cation which undergoes an intramolecular 4+3 cycloaddition.

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