Artigo Acesso aberto Revisado por pares

Synthetic Biology of Proteins: Tuning GFPs Folding and Stability with Fluoroproline

2008; Public Library of Science; Volume: 3; Issue: 2 Linguagem: Inglês

10.1371/journal.pone.0001680

ISSN

1932-6203

Autores

Thomas Steiner, P. Hess, Jae Hyun Bae, Birgit Wiltschi, Luis Moroder, Nediljko Budiša,

Tópico(s)

Enzyme Structure and Function

Resumo

Proline residues affect protein folding and stability via cis/trans isomerization of peptide bonds and by the C(gamma)-exo or -endo puckering of their pyrrolidine rings. Peptide bond conformation as well as puckering propensity can be manipulated by proper choice of ring substituents, e.g. C(gamma)-fluorination. Synthetic chemistry has routinely exploited ring-substituted proline analogs in order to change, modulate or control folding and stability of peptides.

Referência(s)