Artigo Revisado por pares

Design of Sequence‐Specific DNA‐Binding Ligands

1997; Wiley; Volume: 3; Issue: 4 Linguagem: Inglês

10.1002/chem.19970030404

ISSN

1521-3765

Autores

Peter E. Nielsen,

Tópico(s)

RNA Interference and Gene Delivery

Resumo

Abstract Double‐stranded DNA can be viewed as a multifunctional, modular receptor that can be read sequence‐selectively in a digital way (base pair per base pair) by a complementary, similarly modular ligand. This principle has been exploited in several approaches to design sequence‐specific DNA‐binding ligands, such as triplex‐forming oligonucleotides, peptide nucleic acids and minor groove binding polyamides.

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