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Artigo Revisado por pares
BIBTEX RIS

3,3-Bisaryloxindoles as mineralocorticoid receptor antagonists

2005; Elsevier BV; Volume: 15; Issue: 10 Linguagem: Inglês

10.1016/j.bmcl.2005.03.086

ISSN

1464-3405

Autores

David A. Neel, Matthew L. Brown, Peter A. Lander, Timothy A. Grese, Jean Defauw, Robert A. Doti, Todd Fields, Sally Ann Kelley, Stephon C. Smith, Karen M. Zimmerman, Mitchell I. Steinberg, Prabhakar K. Jadhav,

Tópico(s)

ATP Synthase and ATPases Research

Resumo

Syntheses and SAR studies of 3,3-bisaryloxindole analogues provided potent mineralocorticoid receptor (MR) antagonists that were selective over other steroid nuclear hormone receptors.

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