Editorial Acesso aberto Revisado por pares

Harnessing dynamic combinatorial chemistry in the search for new ligands for protein targets

2015; Future Science Ltd; Volume: 7; Issue: 16 Linguagem: Inglês

10.4155/fmc.15.146

ISSN

1756-8927

Autores

Leticia Monjas, Anna K. H. Hirsch,

Tópico(s)

Supramolecular Chemistry and Complexes

Resumo

Future Medicinal ChemistryVol. 7, No. 16 EditorialHarnessing dynamic combinatorial chemistry in the search for new ligands for protein targetsLeticia Monjas & Anna KH HirschLeticia Monjas Stratingh Institute for Chemistry, University of Groningen, Nijenborgh 7, 9747AG, Groningen, The NetherlandsSearch for more papers by this author & Anna KH Hirsch*Author for correspondence: E-mail Address: a.k.h.hirsch@rug.nl Stratingh Institute for Chemistry, University of Groningen, Nijenborgh 7, 9747AG, Groningen, The NetherlandsSearch for more papers by this authorPublished Online:29 Oct 2015https://doi.org/10.4155/fmc.15.146AboutSectionsView ArticleView Full TextPDF/EPUB ToolsAdd to favoritesDownload CitationsTrack CitationsPermissionsReprints ShareShare onFacebookTwitterLinkedInRedditEmail View articleKeywords: drug discoverydynamic combinatorial chemistryinhibitorsmolecular recognitionReferences1 Huc I, Lehn J-M. 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ChemMedChem 7, 1678–1690 (2012).Crossref, Medline, CAS, Google ScholarFiguresReferencesRelatedDetailsCited ByAssembly of split aptamers by dynamic pH-responsive covalent ligation1 January 2023 | Chemical Communications, Vol. 59, No. 38Identification and synthesis of selective cholesterol esterase inhibitor using dynamic combinatorial chemistryBioorganic Chemistry, Vol. 119Contemporary medicinal-chemistry strategies for the discovery of selective butyrylcholinesterase inhibitorsDrug Discovery Today, Vol. 24, No. 2Dynamic Combinatorial Chemistry: A New Methodology Comes of Age11 December 2018 | Chemistry – A European Journal, Vol. 25, No. 1Analytical Methods in Protein-Templated Dynamic Combinatorial ChemistryThe ways and means of fragment-based drug designPharmacology & Therapeutics, Vol. 167Combinatorial Chemistry Online Volume 18, Issue 2, February 2016Combinatorial Chemistry - an Online Journal, Vol. 18, No. 2Advances at the intersection of chemical biology and medicinal chemistryAli Tavassoli16 November 2015 | Future Medicinal Chemistry, Vol. 7, No. 16 Vol. 7, No. 16 STAY CONNECTED Metrics Downloaded 113 times History Published online 29 October 2015 Published in print October 2015 Information© Future Science LtdKeywordsdrug discoverydynamic combinatorial chemistryinhibitorsmolecular recognitionFinancial & competing interests disclosureThe authors have no relevant affiliations or financial involvement with any organization or entity with a financial interest in or financial conflict with the subject matter or materials discussed in the manuscript. This includes employment, consultancies, honoraria, stock ownership or options, expert testimony, grants or patents received or pending, or royalties.No writing assistance was utilized in the production of this manuscript.PDF download

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