Artigo Revisado por pares

Ytterbium(III) Triflate/TMSCl: Efficient Catalyst for Imino Ene Reaction

1999; American Chemical Society; Volume: 2; Issue: 2 Linguagem: Inglês

10.1021/ol991260s

ISSN

1523-7060

Autores

Masamichi Yamanaka, Atsushi Nishida, Masako Nakagawa,

Tópico(s)

Synthesis and Reactivity of Heterocycles

Resumo

[reaction: see text] Ytterbium trifluoromethanesulfonate [Yb(OTf)3] catalyzed the imino ene reaction of N-tosyl aldimine with alpha-methylstyrene to give a homoallylamine in moderate yield. Furthermore, addition of a catalytic amount of chlorotrimethylsilane (TMSCI) dramatically enhanced the imino ene reaction.

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