Methyl 2-((Succinimidooxy)carbonyl)benzoate (MSB): A New, Efficient Reagent for N -Phthaloylation of Amino Acid and Peptide Derivatives
2002; American Chemical Society; Volume: 67; Issue: 11 Linguagem: Inglês
10.1021/jo016347h
ISSN1520-6904
AutoresJ. Richard Casimir, Gilles Guichard, Jean‐Paul Briand,
Tópico(s)Fluorine in Organic Chemistry
ResumoA new, efficient, and readily available reagent, methyl 2-((succinimidooxy)carbonyl)benzoate (MSB), for N-phthaloylation of amino acids and amino acid derivatives is described. The phthaloylation procedure is simple and racemization-free and gives excellent results with α-amino acids, α-amino alcohols, dipeptides, α-amino carboxamides, and α-amino esters.
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