Artigo Acesso aberto Revisado por pares

A caged E3 ligase ligand for PROTAC-mediated protein degradation with light

2020; Royal Society of Chemistry; Volume: 56; Issue: 41 Linguagem: Inglês

10.1039/d0cc00523a

ISSN

1364-548X

Autores

Cyrille S. Kounde, Maria M. Shchepinova, Charlie N. Saunders, Marcel Muelbaier, M.D. Rackham, John D. Harling, Edward W. Tate,

Tópico(s)

Peptidase Inhibition and Analysis

Resumo

Caging of a widely used Von Hippel Lindau E3 ligase ligand for targeted protein degradation with PROTACs allows light-activated proteolysis.

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