Discovery of spirohydantoins as selective, orally bioavailable inhibitors of p300/CBP histone acetyltransferases
2021; Elsevier BV; Volume: 39; Linguagem: Inglês
10.1016/j.bmcl.2021.127854
ISSN1464-3405
AutoresZhiqin Ji, Richard F. Clark, Vikram Bhat, Terkel Hansen, Loren Lasko, Kenneth D. Bromberg, Vlasios Manaves, Mikkel A. Algire, Ruth L. Martin, Wei Qiu, Maricel Torrent, Clarissa G. Jakob, Hong Liu, Philip A. Cole, Ronen Marmorstein, Edward A. Kesicki, Albert Lai, Michael R. Michaelides,
Tópico(s)Genomics and Chromatin Dynamics
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