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Organocatalytic Regio‐ and Stereoselective Inverse‐Electron‐Demand Aza‐Diels–Alder Reaction of α,β‐Unsaturated Aldehydes and N ‐Tosyl‐1‐aza‐1,3‐butadienes

2009; Wiley; Volume: 121; Issue: 30 Linguagem: Inglês

10.1002/ange.200902216

1521-3757

Bo Han, Zhao‐Quan He, Jun‐Long Li, Rui Li, Kun Jiang, Tian‐Yu Liu, Ying‐Chun Chen,

Chemical Synthesis and Analysis

Angewandte ChemieVolume 121, Issue 30 p. 5582-5585 Zuschrift Organocatalytic Regio- and Stereoselective Inverse-Electron-Demand Aza-Diels–Alder Reaction of α,β-Unsaturated Aldehydes and N-Tosyl-1-aza-1,3-butadienes† Bo Han, Bo Han Key Laboratory of Drug-Targeting and Drug-Delivery Systems of the Education Ministry, Department of Medicinal Chemistry, West China School of Pharmacy, Sichuan University, Chengdu, 610041 (China), Fax: (+86) 28-8550-2609Search for more papers by this authorZhao-Quan He, Zhao-Quan He Key Laboratory of Drug-Targeting and Drug-Delivery Systems of the Education Ministry, Department of Medicinal Chemistry, West China School of Pharmacy, Sichuan University, Chengdu, 610041 (China), Fax: (+86) 28-8550-2609Search for more papers by this authorJun-Long Li, Jun-Long Li Key Laboratory of Drug-Targeting and Drug-Delivery Systems of the Education Ministry, Department of Medicinal Chemistry, West China School of Pharmacy, Sichuan University, Chengdu, 610041 (China), Fax: (+86) 28-8550-2609Search for more papers by this authorRui Li Dr., Rui Li Dr. State Key Laboratory of Biotherapy, West China Hospital, Sichuan University, Chengdu, 610041 (China)Search for more papers by this authorKun Jiang, Kun Jiang Key Laboratory of Drug-Targeting and Drug-Delivery Systems of the Education Ministry, Department of Medicinal Chemistry, West China School of Pharmacy, Sichuan University, Chengdu, 610041 (China), Fax: (+86) 28-8550-2609Search for more papers by this authorTian-Yu Liu Dr., Tian-Yu Liu Dr. Key Laboratory of Drug-Targeting and Drug-Delivery Systems of the Education Ministry, Department of Medicinal Chemistry, West China School of Pharmacy, Sichuan University, Chengdu, 610041 (China), Fax: (+86) 28-8550-2609Search for more papers by this authorYing-Chun Chen Prof. Dr., Ying-Chun Chen Prof. Dr. ycchenhuaxi@yahoo.com.cn Key Laboratory of Drug-Targeting and Drug-Delivery Systems of the Education Ministry, Department of Medicinal Chemistry, West China School of Pharmacy, Sichuan University, Chengdu, 610041 (China), Fax: (+86) 28-8550-2609 State Key Laboratory of Biotherapy, West China Hospital, Sichuan University, Chengdu, 610041 (China)Search for more papers by this author Bo Han, Bo Han Key Laboratory of Drug-Targeting and Drug-Delivery Systems of the Education Ministry, Department of Medicinal Chemistry, West China School of Pharmacy, Sichuan University, Chengdu, 610041 (China), Fax: (+86) 28-8550-2609Search for more papers by this authorZhao-Quan He, Zhao-Quan He Key Laboratory of Drug-Targeting and Drug-Delivery Systems of the Education Ministry, Department of Medicinal Chemistry, West China School of Pharmacy, Sichuan University, Chengdu, 610041 (China), Fax: (+86) 28-8550-2609Search for more papers by this authorJun-Long Li, Jun-Long Li Key Laboratory of Drug-Targeting and Drug-Delivery Systems of the Education Ministry, Department of Medicinal Chemistry, West China School of Pharmacy, Sichuan University, Chengdu, 610041 (China), Fax: (+86) 28-8550-2609Search for more papers by this authorRui Li Dr., Rui Li Dr. State Key Laboratory of Biotherapy, West China Hospital, Sichuan University, Chengdu, 610041 (China)Search for more papers by this authorKun Jiang, Kun Jiang Key Laboratory of Drug-Targeting and Drug-Delivery Systems of the Education Ministry, Department of Medicinal Chemistry, West China School of Pharmacy, Sichuan University, Chengdu, 610041 (China), Fax: (+86) 28-8550-2609Search for more papers by this authorTian-Yu Liu Dr., Tian-Yu Liu Dr. Key Laboratory of Drug-Targeting and Drug-Delivery Systems of the Education Ministry, Department of Medicinal Chemistry, West China School of Pharmacy, Sichuan University, Chengdu, 610041 (China), Fax: (+86) 28-8550-2609Search for more papers by this authorYing-Chun Chen Prof. Dr., Ying-Chun Chen Prof. Dr. ycchenhuaxi@yahoo.com.cn Key Laboratory of Drug-Targeting and Drug-Delivery Systems of the Education Ministry, Department of Medicinal Chemistry, West China School of Pharmacy, Sichuan University, Chengdu, 610041 (China), Fax: (+86) 28-8550-2609 State Key Laboratory of Biotherapy, West China Hospital, Sichuan University, Chengdu, 610041 (China)Search for more papers by this author First published: 08 July 2009 https://doi.org/10.1002/ange.200902216Citations: 98 † We are grateful for the financial support of the NSFC (20772084) and Sichuan Province Government (07ZQ026-027). Read the full textAboutPDF ToolsRequest permissionAdd to favorites ShareShare Give accessShare full text accessShare full-text accessPlease review our Terms and Conditions of Use and check box below to share full-text version of article.I have read and accept the Wiley Online Library Terms and Conditions of UseShareable LinkUse the link below to share a full-text version of this article with your friends and colleagues. Learn more.Copy URL Share a linkShare onFacebookTwitterLinkedInRedditWechat Graphical Abstract Dienamine, die in situ aus einem chiralen sekundären Amin und einem α,β-ungesättigten Aldehyd entstehen, liefern in der α-regioselektiven Titelreaktion mit ausgezeichneter Enantioselektivität hochfunktionalisierte Piperidinderivate (siehe Schema). Die Produkte ließen sich in eine Vielzahl nützlicher cyclischer Gerüste überführen. Ts=4-Toluolsulfonyl. Citing Literature Supporting Information Detailed facts of importance to specialist readers are published as "Supporting Information". Such documents are peer-reviewed, but not copy-edited or typeset. They are made available as submitted by the authors. Filename Description ange_200902216_sm_miscellaneous_information.pdf13.4 MB miscellaneous information Please note: The publisher is not responsible for the content or functionality of any supporting information supplied by the authors. Any queries (other than missing content) should be directed to the corresponding author for the article. Volume121, Issue30July 13, 2009Pages 5582-5585 This is the German version of Angewandte Chemie. Note for articles published since 1962: Do not cite this version alone. Take me to the International Edition version with citable page numbers, DOI, and citation export. We apologize for the inconvenience. RelatedInformation